反应条件
Multi-step reaction with 3 steps 1: 40.05 g / aq. HCl / 48 h / Ambient temperature2: 10 percent / HCl / methanol / 5 deg C, 3 h -> room temperature, 18 h3: 82 percent / LiAlH4 / tetrahydrofuran
参考文献
Saunders, John; Showell, Graham A.; Snow, Roger J; Baker, Raymond; Harley, Elizabeth A.; Freedman, Stephen B. Journal of Medicinal Chemistry, 1988 , vol. 31, # 2 p. 486 - 491