反应条件
1: (dimethylamino)pyridine / pyridine / 0.17 h / Ambient temperature
2: 1.) trimethylsilyl chloride, NaI, 2.) triethylamine / 1.) acetonitrile, benzonitrile, 65 deg C, 45 min, reflux, 15 min
View Scheme
参考文献
Warpehoski; Gebhard; Kelly; Krueger; Li; McGovren; Prairie; Wicnienski; Wierenga
Journal of Medicinal Chemistry, 1988 , vol. 31, # 3 p. 590 - 603