反应条件
1: 1.) SOCl2, 2.) K2CO3, / 1.) CH2Cl2, 0 to 10 deg C, 1.5 h, 2.) DMF, RT; 18 h,
2: 60 percent / 80percent m-CPBA, / CH2Cl2 / 0.5 h
View Scheme
参考文献
Uchida; Chihiro; Morita; Kanbe; Yamashita; Yamasaki; Yabuuchi; Nakagawa
Chemical and Pharmaceutical Bulletin, 1989 , vol. 37, # 8 p. 2109 - 2116