反应条件
1: 73 percent / dimethylformamide / 15 h / Ambient temperature 2: trifluoroacetic acid; Et3N 3: 71 percent / dimethylformamide / 15 h / Ambient temperature 4: trifluoroacetic acid; Et3N 5: 69 percent / dimethylformamide / 15 h / Ambient temperature 6: trifluoroacetic acid; Et3N 7: 63 percent / dimethylformamide / 48 h / 30 °C 8: 79 percent / hydrogen / Pd View Scheme
参考文献
Kawasaki, Koichi; Tsuji, Toshiki; Maeda, Misuko; Matsumoto, Tatsuya; Hirase, Katsuhiko
Chemical & Pharmaceutical Bulletin, 1987 , vol. 35, # 3 p. 1044 - 1048