6-氟-7-哌嗪-1-甲基-4-氧代-[1,3]硫氮杂环[3,2-a]喹啉-3-羧酸乙酯合成路线 (共 11 条)
反应条件
1: 88 percent / KOH / 2-methyl-propan-2-ol; H2O / 1 h / 50 - 60 °C 2: 62 percent / KHCO3 / dimethylformamide / 5 h / Ambient temperature View Scheme
参考文献
CIPLA LIMITED; PATHI, Srinivas Laxminarayan; RAO, Dharmaraj Ramachandra; KANKAN, Rajendra; CHINIMILLI, Venugopalarao; CURTIS, Philip Anthony
Patent: WO2012/1357 A1, 2012 ;