4-(三氟甲基磺酰氧基)哌啶-1-羧酸叔丁酯合成路线 (共 2 条)
反应条件
triethylamine in dichloromethane T=0°C; 3 h;
参考文献
MERCK FROSST CANADA LTD.
Patent: WO2006/130986 A1, 2006 ;
Location in patent: Page/Page column 37 ;
WO 2006/130986 A1
反应条件
caesium carbonate in N,N-dimethyl-formamide
T=70°C;
参考文献
MERCK FROSST CANADA LTD.
Patent: WO2006/130986 A1, 2006 ;
Location in patent: Page/Page column 37 ;
WO 2006/130986 A1