1: With N-ethyl-N,N-diisopropylamine in tetrahydrofuran
T=0°C; 0.25 h;
2: With phosphonic acid diethyl ester in tetrahydrofuran
T=20°C; 1 h; Product distribution / selectivity;
参考文献
Bristol-Myers Squibb Company
Patent: US2009/111858 A1, 2009 ;
Location in patent: Page/Page column 6; 18 ;