反应条件
1: With diazomethyl-trimethyl-silane in tetrahydrofuran; diethyl ether; acetonitrile T=0 - 20°C; 2 h; 2: With water; silver(I) acetate in tetrahydrofuran; 1,4-dioxane; diethyl ether; acetonitrile T=100°C; 2 h;
参考文献
TAISHO PHARMACEUTICAL CO., LTD; Kuwada, Takeshi; Yoshinaga, Mitsukane; Ishizaka, Tomoko; Wakasugi, Daisuke; Shirokawa, Shin-ichi; Hattori, Nobutaka; Shimazaki, Youichi; Miyakoshi, Naoki
Patent: US2013/197217 A1, 2013 ;
Location in patent: Paragraph 0523; 0524; 0525 ;