[(1R)-1-(4-氰基苯基)乙基]氨基甲酸叔丁酯合成路线 (共 1 条)
反应条件
1: in N,N-dimethyl-formamide 1 h; 2: With tetrakis(triphenylphosphine) palladium(0) in N,N-dimethyl-formamide T=70 - 75°C; 20.5 h;
参考文献
PFIZER INC.
Patent: WO2009/60278 A1, 2009 ;
Location in patent: Page/Page column 48 ;