反应条件
1: 1.) potassium bis(trimethylsilyl)amide / 1.) DMF, 15 min, 2.) DMF, a) 20 deg C, 3 h, b) 40 deg C, 2 h 2: 73 percent / methanolic NH3 / 18 °C View Scheme
参考文献
Borcherding; Narayanan; Hasobe; McKee; Keller; Borchardt
Journal of Medicinal Chemistry, 1988 , vol. 31, # 9 p. 1729 - 1738
