5-溴-3-碘-4-甲基-2-吡啶胺合成路线 （共 2 条）
反应条件
1: With N-iodo-succinimide; trifluoroacetic acid in acetic acid T=20°C; 2.5 h; 2: With ammonia in water Cooling;
参考文献
Daiichi Sankyo Company, Limited
Patent: US2011/82138 A1, 2011 ;
Location in patent: Page/Page column 32 ;
US 20110082138 A1
反应条件
1: triethylamine; copper(l) iodide / bis-triphenylphosphine-palladium(II) chloride / tetrahydrofuran / 20 °C / Inert atmosphere 2: potassium tert-butylate / 1-methyl-pyrrolidin-2-one / 80 °C View Scheme
参考文献
Daiichi Sankyo Company, Limited
Patent: US2011/82138 A1, 2011 ;
US 20110082138 A1
