5-溴-2,3-二氢-7-氮杂吲哚合成路线 （共 3 条）
反应条件
tetrakis(triphenylphosphine) palladium(0) in dimethyl sulfoxide T=120°C; 4 h;
参考文献
Eisai RandD Management Co., Ltd.
Patent: EP1782811 A1, 2007 ;
Location in patent: Page/Page column 60-61 ;
反应条件
tetrakis(triphenylphosphine) palladium(0); 1,8-diazabicyclo[5.4.0]undec-7-ene in water; tert-butyl alcohol T=85°C; 4 h; Inert atmosphere;
参考文献
Zhang, Dengyou; Sun, Haifeng; Zhang, Lei; Zhou, Yu; Li, Chunpu; Jiang, Hualiang; Chen, Kaixian; Liu, Hong
Chemical Communications, 2012 , vol. 48, # 23 p. 2909 - 2911
反应条件
manganese(IV) oxide in dichloromethane 72 h;
参考文献
EISAI LONDON RESEARCH LABORATORIES LIMITED
Patent: WO2004/78757 A2, 2004 ;
Location in patent: Page 65; 66-67 ;
