4-(6-溴吡啶-2-基)-1,4-二氮杂烷-1-羧酸叔丁酯合成路线 (共 1 条)
反应条件
N-ethyl-N,N-diisopropylamine in ethanol T=100°C; 16 h;
参考文献
F. HOFFMANN-LA ROCHE AG; GENENTECH, INC.; DO, Steven; HU, Huiyong; KOLESNIKOV, Aleksandr; TSUI, Vickie, H.; WANG, Xiaojing
Patent: WO2014/1377 A1, 2014 ;
Location in patent: Page/Page column 103 ;