2,3-二氟-5-(4,4,5,5-四甲基-1,3,2-二噁硼烷-2-基)吡啶合成路线 （共 3 条）
反应条件
potassium acetate; tris-(dibenzylideneacetone)dipalladium(0); tri-cyclo-hexyl-phosphine in 1,4-dioxane T=80°C; 10 h;
参考文献
EP2221301 A1, ;
Page/Page column 44 ;
反应条件
(1,1'-bis(diphenylphosphino)ferrocene)palladium(II) dichloride; potassium acetate in dimethyl sulfoxide T=100°C; Inert atmosphere;
参考文献
WO2013/74387 A1, ;
Page/Page column 43; 44 ;
反应条件
dihydrogen peroxide in tetrahydrofuran; water T=20°C; 2 h;
参考文献
GLAXO GROUP LIMITED; WAN, Zehong; LONG, Kai; SANG, Yingxia; SU, Xiaobo
Patent: WO2013/13503 A1, 2013 ;
Location in patent: Page/Page column 35 ;
WO 2013/013503 A1
