2-(4-氨基-1-(叔丁氧基羰基)哌啶-4-基)乙酸合成路线 (共 1 条)
反应条件
ammonium acetate in butan-1-ol 3 h; Reflux;
参考文献
FIBROGEN, INC.; HO, Wen-Bin; ZHAO, Hongda; DENG, Shaojiang; NG, Danny; WRIGHT, Lee R.; WU, Min; ZHOU, Xiaoti; AREND, Michael P.; FLIPPIN, Lee A.
Patent: WO2013/134660 A1, 2013 ;
Location in patent: Paragraph 0373 ;