6-(4,4,5,5-四甲基-1,3,2-二噁硼烷-2-基)-[1,2,4]噻唑并[1,5-a]吡啶合成路线 (共 1 条)
反应条件
1: With potassium acetate in 1,4-dioxane 0.25 h; 2: With tri-cyclo-hexyl-phosphine; tris-(dibenzylideneacetone)dipalladium(0) in 1,4-dioxane T=100°C; 2.25 h;
参考文献
WO2009/74812 A1, ;
Page/Page column 36 ;
WO 2009/074812 A1