反应条件
1: 96 percent / DEPC, triethylamine / tetrahydrofuran / 6 h / 0 °C 2: 4N HCl / dioxane / 0.5 h / Ambient temperature 3: 91 percent / DEPC, triethylamine / tetrahydrofuran / 6 h / 0 °C 4: 4N HCl / dioxane / 0.5 h / Ambient temperature 5: 71 percent / DEPC, triethylamine / tetrahydrofuran / 8 h / 0 °C View Scheme
参考文献
Nishi; Saito; Nagahori; Kataoka; Morisawa; Yabe; Sakurai; Higashida; Shoji; Matsushita; Iijima; Ohizumi; Koike
Chemical and Pharmaceutical Bulletin, 1990 , vol. 38, # 1 p. 103 - 109