反应条件
palladium diacetate; potassium carbonate; 2,2'-bis-(diphenylphosphino)-1,1'- binaphthyl in toluene 18 h; Inert atmosphereReflux;
参考文献
Hartz, Richard A.; Ahuja, Vijay T.; Rafalski, Maria; Schmitz, William D.; Brenner, Allison B.; Denhart, Derek J.; Ditta, Jonathan L.; Deskus, Jeffrey A.; Yue, Eddy W.; Arvanitis, Argyrios G.; Lelas, Snjezana; Li, Yu-Wen; Molski, Thaddeus F.; Wong, Harvey; Grace, James E.; Lentz, Kimberley A.; Li, Jianqing; Lodge, Nicholas J.; Zaczek, Robert; Combs, Andrew P.; Olson, Richard E.; Mattson, Ronald J.; Bronson, Joanne J.; Macor, John E.
Journal of Medicinal Chemistry, 2009 , vol. 52, # 14 p. 4161 - 4172