5-硝基-6-三氟甲基-2(1H)-吡啶酮合成路线 (共 1 条)
反应条件
1: trichlorophosphate; N,N-dimethyl-formamide / 16 h / 90 °C 2: iron; ammonium chloride / methanol / 2 h / |Reflux View Scheme
参考文献
PHENEX PHARMACEUTICALS AG; STEENECK, Christoph; KINZEL, Olaf; GEGE, Christian; KLEYMANN, Gerald; HOFFMANN, Thomas
Patent: WO2013/79223 A1, 2013 ;