反应条件
1: 1.) H2S, aq. NaOH, 2.) 15percent H2O2 / 1.) RT 2: 67 percent / POCl3, pyridine / 130 - 140 °C View Scheme
参考文献
Yevich, Joseph P.; New, James S.; Smith, David W.; Lobeck, Walter G.; Catt, John D.; et al.
Journal of Medicinal Chemistry, 1986 , vol. 29, # 3 p. 359 - 369