1: 62 percent / NaH / N,N-dimethyl-acetamide / 0.17 h / 120 °C
2: 48 percent / POCl3 / 0.5 h / Heating
View Scheme
参考文献
Goncalves, Victor; Brannigan, James A.; Whalley, David; Ansell, Keith H.; Saxty, Barbara; Holder, Anthony A.; Wilkinson, Anthony J.; Tate, Edward W.; Leatherbarrow, Robin J.
Journal of Medicinal Chemistry, 2012 , vol. 55, # 7 p. 3578 - 3582