反应条件
1: 1.) lithium bis(trimethylsilyl)amide / 1.) THF, 078 deg C, 2 h, 2.) THF, a) -78 deg C, 1 h, b) RT, 20 h 2: H2SO4, glacial acetic acid / 1 h / 95 - 100 °C 3: 90 percent / nitric acid, conc. sulfuric acid / 3 h / Ambient temperature View Scheme
参考文献
Cushman, Mark; Zhu, Helen; Geahlen, Robert L.; Kraker, Alan J.
Journal of Medicinal Chemistry, 1994 , vol. 37, # 20 p. 3353 - 3362
