反应条件
sodium acetate; (1,1'-bis(diphenylphosphino)ferrocene)palladium(II) dichloride in N,N-dimethyl-formamide T=80°C; Inert atmosphere;
参考文献
TAKEDA PHARMACEUTICAL COMPANY LIMITED; FENG, Jun; KEUNG, Walter; LARDY, Matthew
Patent: WO2010/129848 A2, 2010 ;
Location in patent: Page/Page column 24-25 ;
WO 2010/129848 A2