2-吗啉-2-(2-(三氟甲基)嘧啶-5-基)乙胺合成路线 (共 2 条)
反应条件
1.1: DIBAL-h / toluene; dichloromethane / 3 h / -78 °C 1.2: 20 °C 2.1: sodium acetate / acetic acid / 20 °C 3.1: ammonium hydroxide; hydrogen / methanol / 0.42 h / 20 °C / 1551.49 Torr / |Inert atmosphere View Scheme
反应条件
1: sodium acetate / acetic acid / 20 °C 2: ammonium hydroxide; hydrogen / methanol / 0.42 h / 20 °C / 1551.49 Torr / |Inert atmosphere View Scheme