反应条件
1: 100 percent / 1 N NaOH / tetrahydrofuran / Heating 2: 1.) 1,1-carbonyldiimidazole / 1.) THF, 1 h View Scheme
参考文献
Musser, John H.; Kreft, Anthony F.; Bender, Reinhold H. W.; Kubrak, Dennis M.; Grimes, David; et al.
Journal of Medicinal Chemistry, 1990 , vol. 33, # 1 p. 240 - 245