2,4-二氨基-5-氟喹唑啉合成路线 (共 3 条)
反应条件
in N,N-dimethyl acetamide T=140 - 142°C; 5 h;
参考文献
Hynes, John B.; Pathak, Alpana; Panos, Constantina H.; Okeke, Claudia C.
Journal of Heterocyclic Chemistry, 1988 , vol. 25, p. 1173 - 1177
反应条件
in diethylene glycol dimethyl ether T=130 - 140°C; 3 h;
参考文献
Harris, Neil V.; Smith, Christopher; Bowden, Keith
Journal of Medicinal Chemistry, 1990 , vol. 33, # 1 p. 434 - 444
反应条件
in N,N-dimethyl-formamide T=135°C; 6 h;
参考文献
Journal of Heterocyclic Chemistry, , vol. 29, # 4 p. 915 - 920