反应条件
1: 80 percent / Cs2CO3 / N,N-dimethyl-acetamide / 24 h / Ambient temperature 2: 79 percent / N,N-dimethyl-acetamide / 6 h / 140 - 142 °C View Scheme
参考文献
Chao, Bo; Tong, Xian-Kun; Tang, Wei; Li, De-Wen; He, Pei-Lan; Garcia, Jean-Michel; Zeng, Li-Min; Gao, An-Hui; Yang, Li; Li, Jia; Nan, Fa-Jun; Jacobs, Michael; Altmeyer, Ralf; Zuo, Jian-Ping; Hu, You-Hong
Journal of Medicinal Chemistry, 2012 , vol. 55, # 7 p. 3135 - 3143