4-氯-5-(三氟甲基)-1H-吡咯并[2,3-B]吡啶-3-胺合成路线 (共 1 条)
反应条件
1: With hydrogenchloride; SnCl2·2H2O in water T=0 - 20°C; 2 h; 2: With sodium hydroxide in water pH=8;
参考文献
ARRAY BIOPHARMA INC.
Patent: WO2009/140320 A1, 2009 ;
Location in patent: Page/Page column 99 ;
WO 2009/140320 A1