反应条件
1: 1) NaH / 1) DMF, 60-70 deg C, 1 h, 2) 80 deg C, overnight 2: NaOH / ethanol; H2O / 2 h / Heating View Scheme
参考文献
DeRuiter, Jack; Swearingen, Blake E.; Wandrekar, Vinay; Mayfield, Charles A.
Journal of Medicinal Chemistry, 1989 , vol. 32, # 5 p. 1033 - 1038