反应条件
(N,N-Dimethylamino)sulfur trifluoride; ammonia 1) CHCl3, 55 deg C, 2.5-3 h, 2) MeOH, r.t., 2.5 h; Yield given. Multistep reaction. Yields of byproduct given;
参考文献
Sufrin, Janice R.; Spiess, Arthur J.; Kramer, Debora L.; Libby, Paul R.; Porter, Carl W.
Journal of Medicinal Chemistry, 1989 , vol. 32, # 5 p. 997 - 1001