反应条件
Multi-step reaction with 2 steps 1: 84 percent / POCl3, N,N-diethylaniline / 2 h / Ambient temperature2: 91 percent / Et3N, H2 / Pd-C / benzene
参考文献
Katagiri; Watanabe; Kaneko Chemical and Pharmaceutical Bulletin, 1988 , vol. 36, # 9 p. 3354 - 3372