3-溴吡唑并[1,5-a]嘧啶-5(4h)-酮合成路线 (共 1 条)
反应条件
N-bromosuccinmide in dichloromethane; N,N-dimethyl-formamide T=20°C; 17 h;
参考文献
ARRAY BIOPHARMA INC.; ANDREWS, Steven W.; CONDROSKI, Kevin Ronald; DE MEESE, Lisa A.; FELL, Jay Bradford; FISCHER, John P.; LE HUEROU, Yvan; JOSEY, John A.; KOCH, Kevin; MIKNIS, Gregory F.; RODRIGUEZ, Martha E.; TOPALOV, George T.; WALLACE, Eli M.; XU, Rui
Patent: WO2011/29027 A1, 2011 ;
Location in patent: Page/Page column 45 ;
WO 2011/029027 A1