反应条件
1: 59 percent / K2CO3, Cu2Br2, N-methyl-2-pyrrolidinone 2: 1.) N-chlorosuccinimide, 2.) glacial acetic acid, 85percent H3PO4 / 1.) CH2Cl2, 2.) reflux View Scheme
参考文献
Sarges, Reinhard; Howard, Harry R.; Koe, B. Kenneth; Weissman, Albert
Journal of Medicinal Chemistry, 1989 , vol. 32, # 2 p. 437 - 444