4-(2,4,6-三氟苯甲酰基)-1H-吡咯-2-羧酸合成路线 (共 1 条)
反应条件
1: 2,4,6-trifluorobenzoyl chloride With AlCl3, aluminium chloride in dichloromethane T=20°C; 0.25 h; Inert atmosphere; 2: pyrrole-2-carboxylic acid ester in dichloromethane T=20°C; 1.16667 h; 3: With hydrogenchloride; water in dichloromethane pH=1;
参考文献
WO2009/152072 A1, ;
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