5-(甲基磺酰胺)吡啶-3-硼酸频那醇酯合成路线 (共 1 条)
反应条件
potassium acetate; (1,1'-bis(diphenylphosphino)ferrocene)palladium(II) dichloride in 1,4-dioxane T=85°C; 8 h; Inert atmosphere;
参考文献
PROGENICS PHARMACEUTICALS, INC.
Patent: WO2009/155527 A2, 2009 ;
Location in patent: Page/Page column 136-137 ;
WO 2009/155527 A2