3-甲基-1H-吡咯并[2,3-B]吡啶-2-羧酸合成路线 (共 1 条)
反应条件
potassium phosphate; magnesium sulfate; acetic acid; Pd0(tris(tert-butyl)phosphine)2 in isobutyramide
T=140°C;
参考文献
IRONWOOD PHARMACEUTICALS INCORPORATED; LUDRIGAN, Regina; JEFFREY, John; MERMERIAN, Ara
Patent: WO2010/5528 A2, 2010 ;
Location in patent: Page/Page column 89-90 ;