5-(叔丁氧基羰基)-2-碘噻唑-4-羧酸乙酯合成路线 (共 1 条)
反应条件
N-iodo-succinimide in N,N-dimethyl-formamide T=60°C; 54 h;
参考文献
MERCK and CO., INC.; MACHACEK, Michelle, R.; HAIDLE, Andrew; ZABIEREK, Anna, A.; KONRAD, Kaleen, M.; ALTMAN, Michael, D.
Patent: WO2010/11375 A2, 2010 ;
Location in patent: Page/Page column 64 ;
WO 2010/011375 A2