Multi-step reaction with 3 steps 1: acetic acid; sodium tris(acetoxy)borohydride / dichloromethane / 1 h / 20 °C2: sodium hydrogencarbonate / dichloromethane / 1 h / 20 °C3: hydrazine / acetonitrile / 24 h / 85 °C
参考文献
RUTGERS, THE STATE UNIVERSITY OF NEW JERSEY; THE BROAD INSTITUTE, INC.; HU, Longqin; MAGESH, Sadagopan; CHEN, Lin; LEWIS, Timothy; MUNOZ, Ben; WANG, Lili Patent: WO2013/67036 A1, 2013 ;