反应条件
1: N-ethyl-N,N-diisopropylamine; HATU / N,N-dimethyl-formamide / 2 h / 0 °C 2: lithium aluminium tetrahydride / diethyl ether / 0.25 h / 0 °C View Scheme
参考文献
MEDIVIR UK LIMITED; AYESA, Susana; ERSMARK, Karolina; GRABOWSKA, Urszula; HEWITT, Ellen; JOeNSSON, Daniel; KAHNBERG, Pia; KLASSON, Bjoern; LIND, Peter; LUNDGREN, Stina; ODEN, Lourdes; PARKES, Kevin; WIKTELIUS, Daniel
Patent: WO2011/70539 A1, 2011 ;
WO 2011/070539 A1
Title/Abstract Full Text Show Details
MEDIVIR UK LIMITED; AYESA, Susana; GRABOWSKA, Urszula; HEWITT, Ellen; JOeNSSON, Daniel; KLASSON, Bjoern; KAHNBERG, Pia; LUNDGREN, Stina; TEJBRANT, Jan; WIKTELIUS, Daniel
Patent: WO2011/158197 A1, 2011 ;
WO 2011/158197 A1