5-(4,4,5,5-四甲基-1,3,2-二噁硼烷-2-基)-吡咯并[2,3-B]吡啶-2(3H)-酮合成路线 (共 1 条)
反应条件
potassium acetate; 1,1'-bis-(diphenylphosphino)ferrocene; (1,1'-bis(diphenylphosphino)ferrocene)palladium(II) dichloride in 1,4-dioxane T=120°C; 8 h;
参考文献
KUDOS PHARMACEUTICALS LIMITED
Patent: WO2008/23161 A1, 2008 ;
Location in patent: Page/Page column 111 ;
WO 2008/023161 A1