反应条件
1: potassium carbonate / N,N-dimethyl-formamide / 8 h 2: tetrakis(triphenylphosphine) palladium(0) / N,N-dimethyl-formamide / 8 h / 110 °C View Scheme
参考文献
MERCK SHARP and DOHME CORP.; PASTERNAK, Alexander; BLIZZARD, Timothy; CHOBANIAN, Harry; DE JESUS, Reynalda; DING, Fa-Xiang; DONG, Shuzhi; GUDE, Candido; KIM, Dooseop; TANG, Haifeng; WALSH, Shawn; PIO, Barbara; JIANG, Jinlong
Patent: WO2013/28474 A1, 2013 ;