反应条件
1: 63 percent / 5-methyl-2-chloro-3-phenyl-2,3-dihydro-1,3,4,2-oxadiazaphosphole, pyridine / Ambient temperature
2: 1.) LDA / 1.) THF, 0 deg C, 30 min, 2.) THF, from 0 deg C to RT
View Scheme
参考文献
De Las Heras, Maria A.; Vaquero, Juan J.; Garcia Navio, Jose L.; Alvarez-Builla, Julio
Tetrahedron, 1996 , vol. 52, # 45 p. 14297 - 14310