反应条件
thionyl chloride 1.) CH2Cl2, RT, 17 h, 2.) CH2Cl2, toluen, reflux, 2 h; Multistep reaction;
参考文献
Kumazawa, Toshiaki; Yanase, Masashi; Harakawa, Hiroyuki; Obase, Hiroyuki; Shirakura, Shiro; et al.
Journal of Medicinal Chemistry, 1994 , vol. 37, # 6 p. 804 - 810