反应条件
1: oxalyl dichloride / N,N-dimethyl-formamide 2: N,N-dimethyl-formamide / 80 °C 3: sodium tetrahydroborate / THF-d8 (tetrahydrofuran-d8); ethanol / 0 °C View Scheme
参考文献
Ding, Derong; Nickell, Justin R.; Deaciuc, Agripina G.; Penthala, Narsimha Reddy; Dwoskin, Linda P.; Crooks, Peter A.
Bioorganic and Medicinal Chemistry, 2013 , vol. 21, # 21 p. 6771 - 6777