6-溴-2-硝基吡啶-3-胺合成路线 (共 1 条)
反应条件
1: With bromine; sodium acetate in acetic acid 2: With sodium hydrogencarbonate T=0°C; pH=~ 7;
参考文献
ASTRAZENECA AB; BJOeRK, Seth; DELISSER, Vern; JOHNSTROeM, Peter; NILSSON, Nils Anders; RUDA, Katinka; SCHOU, Per Magnus; SWAHN, Britt-Marie
Patent: WO2010/24769 A1, 2010 ;
Location in patent: Page/Page column 31 ;
WO 2010/024769 A1