反应条件
1: 2,2-dimethyl-L-thiazoline-4-carboxylic acid hydrochloride; N-Cbz-glycine fluoride With N-ethyl-N,N-diisopropylamine in N,N-dimethyl-formamide T=20°C; 18 h; 2: methanol With chloro-trimethyl-silane T=20°C; 15 h;
参考文献
Tetrahedron, , vol. 61, # 42 p. 10018 - 10035