反应条件
trimethylsilyl trifluoromethanesulfonate; ammonia; water; bis(trimethyl-silyl)acetamide 1.) acetonitrile, reflux, 2.5 h, 2.) MeOH, 80 deg C, 18 h; Yield given. Multistep reaction. Yields of byproduct given;
参考文献
Robins; Wood; Dalley; Herdewijn; Balzarini; De Clercq
Journal of Medicinal Chemistry, 1989 , vol. 32, # 8 p. 1763 - 1768