2-溴-4-氯-1-(二氟甲氧基)苯合成路线 (共 2 条)
反应条件
water; caesium carbonate in N,N-dimethyl-formamide T=100°C; 16 h;
参考文献
WO2011/3065 A2, ;
Page/Page column 99 ;
WO 2011/003065 A2
反应条件
potassium hydroxide in dichloromethane; water T=0°C; 0.5 h;
参考文献
Angewandte Chemie - International Edition, , vol. 52, # 47 p. 12390 - 12394
Angew. Chem., , vol. 125, # 47 p. 12616 - 12620,5