4-甲基-1,4-苯并噁嗪-3-酮-6-硼酸频那醇酯合成路线 (共 3 条)
反应条件
potassium acetate; 1,1'-bis(di-tert-butylphosphino)ferrocene palladium dichloride in water; acetonitrile T=85°C; 18 h; Inert atmosphere of nitrogen;
参考文献
ASTRAZENECA AB; ASTRAZENECA UK LIMITED; FORD, Rhonan; METE, Antonio; MATHER, Andrew; MILLICHIP, Ian
Patent: WO2010/128324 A1, 2010 ;
Location in patent: Page/Page column 71 ;
WO 2010/128324 A1
参考文献
Incyte Corporation; Zhuo, Jincong; Xu, Meizhong; Qian, Ding-Quan
Patent: US2014/171405 A1, 2014 ;
Location in patent: Page/Page column ;
反应条件
1: water; N,N-dimethyl-formamide View Scheme
参考文献
Incyte Corporation; Zhuo, Jincong; Xu, Meizhong; Qian, Ding-Quan
Patent: US2014/171405 A1, 2014 ;