1: With water; lithium hydroxide hydrate in tetrahydrofuran T=20°C; 3 h; 2: With hydrogenchloride in water pH=3;
参考文献
PHENOMIX CORPORATION; BETANCORT, Juan Manuel; HEPPERLE, Michael E.; CAMPBELL, David Alan; WINN, David T.
Patent: WO2010/33466 A1, 2010 ;
Location in patent: Page/Page column 65-66 ;
WO 2010/033466 A1